Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

David Sedlák; Tyler A. Wilson; Werner Tjarks; Hanna S. Radomska; Hongyan Wang; Jayaprakash Narayana Kolla; Zbigniew J. Leśnikowski; Alena Špičáková; Tehane Ali; Keisuke Ishita; Liva Harinantenaina Rakotondraibe; Sandip Vibhute; Dasheng Wang; Pavel Anzenbacher; Chad Bennett; Petr Bartunek; Christopher C. Coss

doi:10.1021/acs.jmedchem.1c00555

Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

David Sedlák
, Tyler A. Wilson
, Werner Tjarks
, Hanna S. Radomska
, Hongyan Wang
, Jayaprakash Narayana Kolla
, Zbigniew J. Leśnikowski
, Alena Špičáková
, Tehane Ali
, Keisuke Ishita
, Liva Harinantenaina Rakotondraibe
, Sandip Vibhute
, Dasheng Wang
, Pavel Anzenbacher
, Chad Bennett
, Petr Bartunek
, Christopher C. Coss

Institute of Molecular Genetics of the Czech Academy of Sciences
The Ohio State University Comprehensive Cancer Center
The Ohio State University
Institute of Medical Biology PAS
Palacký University
Department of Pharmacology

Research output: Contribution to journal › Article › peer-review

Original language	English
Pages (from-to)	9330-9353
Number of pages	24
Journal	Journal of Medicinal Chemistry
Volume	64
Issue number	13
DOIs	https://doi.org/10.1021/acs.jmedchem.1c00555
State	Published - Jul 8 2021
Externally published	Yes

ASJC Scopus Subject Areas

Molecular Medicine
Drug Discovery

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10.1021/acs.jmedchem.1c00555

Cite this

Sedlák, D., Wilson, T. A., Tjarks, W., Radomska, H. S., Wang, H., Kolla, J. N., Leśnikowski, Z. J., Špičáková, A., Ali, T., Ishita, K., Rakotondraibe, L. H., Vibhute, S., Wang, D., Anzenbacher, P., Bennett, C., Bartunek, P., & Coss, C. C. (2021). Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists. Journal of Medicinal Chemistry, 64(13), 9330-9353. https://doi.org/10.1021/acs.jmedchem.1c00555

Sedlák, D, Wilson, TA, Tjarks, W, Radomska, HS, Wang, H, Kolla, JN, Leśnikowski, ZJ, Špičáková, A, Ali, T, Ishita, K, Rakotondraibe, LH, Vibhute, S, Wang, D, Anzenbacher, P, Bennett, C, Bartunek, P & Coss, CC 2021, 'Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists', Journal of Medicinal Chemistry, vol. 64, no. 13, pp. 9330-9353. https://doi.org/10.1021/acs.jmedchem.1c00555

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title = "Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists",

author = "David Sedl{\'a}k and Wilson, \{Tyler A.\} and Werner Tjarks and Radomska, \{Hanna S.\} and Hongyan Wang and Kolla, \{Jayaprakash Narayana\} and Le{\'s}nikowski, \{Zbigniew J.\} and Alena {\v S}pi{\v c}{\'a}kov{\'a} and Tehane Ali and Keisuke Ishita and Rakotondraibe, \{Liva Harinantenaina\} and Sandip Vibhute and Dasheng Wang and Pavel Anzenbacher and Chad Bennett and Petr Bartunek and Coss, \{Christopher C.\}",

note = "Publisher Copyright: {\textcopyright} 2021 The Authors. Published by American Chemical Society.",

year = "2021",

month = jul,

day = "8",

doi = "10.1021/acs.jmedchem.1c00555",

language = "English",

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AU - Sedlák, David

AU - Wilson, Tyler A.

AU - Tjarks, Werner

AU - Radomska, Hanna S.

AU - Wang, Hongyan

AU - Kolla, Jayaprakash Narayana

AU - Leśnikowski, Zbigniew J.

AU - Špičáková, Alena

AU - Ali, Tehane

AU - Ishita, Keisuke

AU - Rakotondraibe, Liva Harinantenaina

AU - Vibhute, Sandip

AU - Wang, Dasheng

AU - Anzenbacher, Pavel

AU - Bennett, Chad

AU - Bartunek, Petr

AU - Coss, Christopher C.

PY - 2021/7/8

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UR - https://www.scopus.com/pages/publications/85110282923

UR - https://www.scopus.com/pages/publications/85110282923#tab=citedBy

U2 - 10.1021/acs.jmedchem.1c00555

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C2 - 34181409

AN - SCOPUS:85110282923

SN - 0022-2623

VL - 64

SP - 9330

EP - 9353

JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

IS - 13

ER -

Structure-Activity Relationship of para-Carborane Selective Estrogen Receptor β Agonists

ASJC Scopus Subject Areas

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